Products

Enzymes for Research, Diagnostic and Industrial Use

EZH2 Inhibitor, EPZ005687

Cat No.
CEI-0475
Description
A potent and selective inhibitor of histone lysine N-methyltransferase EZH2 (Ki = 24 nM). It displays more than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme, EZH1.
Appearance
White to off-white solid
Product Overview
A potent EZH2 inhibitor
CAS No.
1396772-26-1
Molecular Weight
475.6
Purity
>98% by HPLC
Storage
+4 centigrade
Targets
EZH2
Molecular Formula
C 32 H 37 N 6 O 3
Chemical Name
1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide
Solubility
DMSO (10 mg/ml)
Shipping Conditions
Gel pack
Download Datasheet:



Inquiry
Realted Products
Catalog
ProductName
EC No.
CAS No.
Source
Price
CatalogCEI-0473
ProductNameGSK343
EC No.
CAS No.1346704-33-3
Source
CatalogCEI-0474
ProductNameGSK126
EC No.
CAS No.1346574-57-9
Source
CatalogCEI-0476
ProductNameGSK343
EC No.
CAS No.1346704-33-3
Source
CatalogCEI-0477
EC No.
CAS No.102052-95-9
Source
+ See More >>
Online Inquiry
Name:
*Phone:
*E-mail Address:
Country:
Company/Institution:
*Products or Services Interested:
Quantity:
Project Description:
Our Products are Not Intended for Private Therapeutic Use!
*Verification Code:
Please input "enzymes"(case insensitive) as verification code.

Welcome! For price inquiries, please feel free to contact us through the form below through the form on the left side. We will get back to you as soon as possible.

Sitemap  Privacy Policy
Copyright ©2011 - 2017 Creative Enzymes.
Contact Us 45-1 Ramsey Road, Shirley, NY 11967, USA
Email: info@creative-enzymes.com
Tel: 1-631-562-8517 1-631-448-7888
Fax: 1-631-938-8127
Distributors To view the contact information for a specific location, select the desired country: