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GW843682X

Cat No.
CEI-1359
Product Overview
GW843682X is a selective inhibitor of polo-like kinase 1 (PLK1) and polo-like kinase 3 (PLK3) (IC50 values are 2.2 and 9.1 nM respectively). GW843682X displays >100-fold selectivity over 30 other kinases tested including cdk1 and cdk2.GW843682X inhibits proliferation of most tumor cells in vitro and is selective over normal diploid fibroblasts.
CAS No.
660868-91-7
Molecular Weight
477.46
Purity
0.98
Storage
Store at -20°C
Synonyms
GW 843682X; GW843682; GW-843682X
Targets
PLK1/PLK3
Molecular Formula
C22H18F3N3O4S
Chemical Name
5-(5,6-dimethoxybenzimidazol-1-yl)-3-[[2-(trifluoromethyl)phenyl]methoxy]thiophene-2-carboxamide
Solubility
Soluble in DMSO > 10 mM
Shipping Conditions
Evaluation sample solution: ship with blue ice. All other available size: ship with RT, or blue ice upon request
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