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Tie2 kinase inhibitor

Cat No.
CEI-0025
Description
Tie2 kinase inhibitor
CAS No.
948557-43-5
Molecular Weight
439.53
Purity
>99%
Storage
2 years at -20centigrade Powder
Targets
Tie2 kinase
Molecular Formula
C26H21N3O2S
Chemical Name
4-(5-(6-methoxynaphthalen-2-yl)-2-(4-(methylsulfinyl)phenyl)-1H-imidazol-4-yl)pyridine
Solubility
DMSO 35 mg/mL, Water
In vitro
Tie2 kinase inhibitor exhibits a moderate inhibitory activity against Tie2 tyrosine kinase. Tie2 kinase inhibitor also shows moderate cellular activities with IC50 of 232 nM in HEL cells. Furthermore, Tie2 kinase inhibitor has a remarkable selectivity for Tie2 over p38 (IC50=50 uM) and a >10-fold selectivity over VEGFR2, VEGFR3, and PDGFR1beta.
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