AGI-5198

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Cat No.

CEI-0995

Description

AGI-5198 is a selective inhibitor of IDH1 R132H and R132C mutants. It serves as a potent antitumor compound by inducing demethylation of histone H3K9me3 and expression of genes associated with gliogenic differentiation.

Abbr

AGI-5198(IDH1)

Alias

IDCD, IDH, IDP, IDPC, PICD

Appearance

A crystalline solid.

CAS_No

1355326-35-0

Molecular Weight

462.56

Purity

> 95%

Storage

Room temperature for 24 months as powder, +4 centigrade for 2 weeks in DMSO, or −70 centigrade for 6 months in anhydrous DMSO. Keep DMSO stock solutions out of contact with air. Protect from moisture.

Synonyms

IDCD, IDH, IDP, IDPC, PICD

Targets

IDH1, R132H/R132C

IC50

0.07 μM/0.16 μM

Molecular Formula

C27H31FN4O2

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Our Products Cannot Be Used As Medicines Directly For Personal Use.

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