CEP-33779

inquiry

Cat No.

CEI-1142

Description

CEP-33779 is a highly selective, orally active inhibitor for JAK2 with IC50 of 1.8nM in enzyme and 61nM in cell, comparing to the inhibition for JAK3 with IC50 of 150nM.

Abbr

CEP-33779(JAK2, JAK3)

Alias

JTK10, THCYT3

CAS_No

1346168-57-7

Molecular Weight

462.57

Purity

> 95%

Stability

2 years -20 centigrade Powder
1 month -4 centigrade in DMSO
More than one month -80 centigrade in DMSO

Storage

4 centigrade

Synonyms

JTK10, THCYT3

Targets

JAK2, JAK3

IC50

61nM, 150nM

Molecular Formula

C24H26N6O2S

Chemical Name

N-(3-(4-methylpiperazin-1-yl)phenyl)-8-(4-(methylsulfonyl)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine

Solubility

DMSO > 112mg/mL Water >1mg/mL Ethanol > 4mg/mL

Name:

Email *

Phone:*

Company/Institution:

Country or Region:

Quantity:

Services & Products Interested *

Project Description:

Our Products Cannot Be Used As Medicines Directly For Personal Use.

Products

Online Inquiry