CGP60474

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Cat No.

CEI-1276

Product Overview

CGP60474 is a potent inhibitor of cyclin-dependent kinases (CDKs) with IC50 value of 17 nM for CDK1.It is also an inhibitor of Protein Kinase C (PKC). CDKs are a family of protein kinases regulating the cell cycle. PKC plays an important role in signal transductions, cellular proliferation and differentiation. CGP60474 was highly selective for PKC than other serine/threonine and tyrosine kinases and showed competitive kinetics relative to ATP.

CAS_No

164658-13-3

Molecular Weight

355.82

Purity

0.98

Storage

Store at -20°C

Synonyms

CGP-60474; CGP 60474

Targets

CDKs; PKC

Molecular Formula

C18H18ClN5O

Chemical Name

3-[[4-[2-(3-chloroanilino)pyrimidin-4-yl]pyridin-2-yl]amino]propan-1-ol

Solubility

Soluble in DMSO

Shipping Conditions

Evaluation sample solution: ship with blue ice. All other available size: ship with RT, or blue ice upon request

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Project Description:

Our Products Cannot Be Used As Medicines Directly For Personal Use.

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