CID 2745687

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Cat No.

CEI-0596

Description

Cell-permeable. A potent, competitive, and reversible antagonist of the orphan receptor GPR35 (Ki = 12.8 nM). Prevents the GPR35-mediated increase in ERK1/2 phosphorylation and β-arrestin recruitment induced by pamoic acid.

Appearance

Yellow solid

Product Overview

A potent and reversible antagonist of the orphan receptor GPR36

CAS_No

264233-05-8

Molecular Weight

259.33

Purity

>98% by TLC

Storage

-20 centigrade

Targets

GPR35

Molecular Formula

C₁₇H₁₉F₂N₅O₂S

Chemical Name

Methyl -5-((2-t-butylcarbamothioyl)hydrazono)methyl)-1-(2,4-difluorophenyl)-1H-pyrazole-4-carboxylate

Solubility

DMSO (~25 mg/ml) or EtOH (~ 6 mg/ml)

Shipping Conditions

Gel pack

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Project Description:

Our Products Cannot Be Used As Medicines Directly For Personal Use.

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