PFI-1

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Cat No.

CEI-0408

Description

PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC50 values of 98 nM and 0.22 μM, respectively.

Appearance

Crystalline solid

Product Overview

A potent BET bromodomain inhibitor

CAS_No

1403764-72-6

Molecular Weight

358.48

Purity

>98%

Storage

-20 centigrade

Targets

BRD2, BRD4

Molecular Formula

C 16 H 17 N 3 O 4 S

Chemical Name

2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide

Solubility

DMSO

Shipping Conditions

Gel Pack

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Project Description:

For research and industrial use only, not for personal medicinal use.

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