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C646, p300/CBP Inhibitor

Cat No.
CEI-0599
Description
Cell-permeable. A reversible, p300/CBP (CREB-binding protein) histone acetyltransferase (HAT) inhibitor (Ki = 400 nM). Specific inhibition to p300 (86%) compared to N-acetyltransferase, PCAF, GCN5, Rtt109, Sas or MOZ histone acetyltransferases (<10%). Suppresses histone H3 and H4 acetylation in mouse fibroblast cell lines.
Appearance
White solid
Product Overview
A reversible, p300/CBP (CREB-binding protein) histone acetyltransferase (HAT) inhibitor
CAS No.
328968-36-1
Molecular Weight
503
Purity
>98% by TLC
Storage
-20 centigrade
Targets
EP300, CREBBP
Molecular Formula
C₂₄H₁₉N₃O₆
Chemical Name
(E)-4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)-methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid
Solubility
DMSO
Shipping Conditions
Gel pack
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