Products

Enzymes for Research, Diagnostic and Industrial Use

GSK343

Cat No.
CEI-0473
Description
A potent histone H3-lysine 27 (H3K27) methyltransferase EZH2 inhibitor (IC50 = 4 nM). Diplays 1000-fold selectivity for other HMTs except EZH1 (60-fold selectivity). GSK343 inhibits H3K27 methylation in HCC1806 cells with an IC50 of
Appearance
Liquid
Product Overview
A potent EZH2 inhibitor
CAS No.
1346704-33-3
Molecular Weight
652.7
Purity
>95% by HPLC
Storage
-20 centigrade
Targets
EZH2
Molecular Formula
C 31 H 39 N 7 O 2
Chemical Name
1-Isopropyl-N-((6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl)-6-(2-(4-methylpiperazin-1-yl)pyridine-4-yl)-1H-indazole-4-carboxamide
Shipping Conditions
Gel pack
Download Datasheet:



Inquiry
Realted Products
Catalog
ProductName
EC No.
CAS No.
Source
Price
CatalogCEI-0474
ProductNameGSK126
EC No.
CAS No.1346574-57-9
Source
CatalogCEI-0475
EC No.
CAS No.1396772-26-1
Source
CatalogCEI-0476
ProductNameGSK343
EC No.
CAS No.1346704-33-3
Source
CatalogCEI-0477
EC No.
CAS No.102052-95-9
Source
+ See More >>
Online Inquiry
Name:
*Phone:
*E-mail Address:
Country:
Company/Institution:
*Products or Services Interested:
Quantity:
Project Description:
Our Products are Not Intended for Private Therapeutic Use!
*Verification Code:
Please input "enzymes"(case insensitive) as verification code.

Welcome! For price inquiries, please feel free to contact us through the form below through the form on the left side. We will get back to you as soon as possible.

Sitemap  Privacy Policy
Copyright ©2011 - 2017 Creative Enzymes.
Contact Us 45-1 Ramsey Road, Shirley, NY 11967, USA
Email: info@creative-enzymes.com
Tel: 1-631-562-8517 1-631-448-7888
Fax: 1-631-938-8127
Distributors To view the contact information for a specific location, select the desired country: